Synthesis of C-8 methanesulphonate substituted pyrrolobenzodiazepines as potential antitumour agents.
نویسندگان
چکیده
The facile synthesis of C-8 methanesulphonate substituted pyrrolobenzodiazepines is described. These have been prepared by linking the methanesulphonate at C-8 position with alkanol spacer and their in vitro cytotoxicity have been described.
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ورودعنوان ژورنال:
- Bioorganic & medicinal chemistry letters
دوره 13 20 شماره
صفحات -
تاریخ انتشار 2003